{"id":39635,"date":"2026-01-28T22:26:24","date_gmt":"2026-01-28T21:26:24","guid":{"rendered":"https:\/\/europa-peptide.com\/?post_type=product&#038;p=39635"},"modified":"2026-06-14T00:40:23","modified_gmt":"2026-06-13T22:40:23","slug":"pt-141-10mg","status":"publish","type":"product","link":"https:\/\/europa-peptide.com\/de\/shop\/pt-141-10mg\/","title":{"rendered":"PT-141 10mg"},"content":{"rendered":"<p data-start=\"151\" data-end=\"220\"><strong data-start=\"151\" data-end=\"220\">PT-141 (Bremelanotid) - Peptid zur Modulation des Melanocortin-Rezeptors<\/strong><\/p>\n<p data-start=\"222\" data-end=\"494\"><strong data-start=\"222\" data-end=\"238\">Zusammensetzung:<\/strong> PT-141 (10 mg lyophilisiertes Peptidpulver)<br data-start=\"280\" data-end=\"283\" \/><strong data-start=\"283\" data-end=\"296\">Kategorie:<\/strong> Peptid<br data-start=\"304\" data-end=\"307\" \/><strong data-start=\"307\" data-end=\"316\">Form:<\/strong> 10 mg Fl\u00e4schchen mit gefriergetrocknetem Pulver<br data-start=\"352\" data-end=\"355\" \/><strong data-start=\"355\" data-end=\"374\">Verwaltung:<\/strong> Subkutane Forschungsanwendung nach Rekonstitution mit sterilem oder bakteriostatischem Wasser (je nach Studiendesign)<\/p>\n<hr data-start=\"496\" data-end=\"499\" \/>\n<h3 data-start=\"501\" data-end=\"520\">Was ist PT-141?<\/h3>\n<p data-start=\"522\" data-end=\"738\">PT-141, auch bekannt als <strong data-start=\"544\" data-end=\"561\">Bremelanotid<\/strong>, ist ein synthetisches Peptid, das von Melanocortin-Analoga abgeleitet ist und speziell f\u00fcr die Interaktion mit <strong data-start=\"668\" data-end=\"707\">Melanocortin-Rezeptoren (MC3R, MC4R)<\/strong> im zentralen Nervensystem.<\/p>\n<p data-start=\"740\" data-end=\"959\">Im Gegensatz zu Peptiden, die \u00fcber hormonelle oder vaskul\u00e4re Pfade wirken, wurde PT-141 auf seine <strong data-start=\"836\" data-end=\"878\">direkte Aktivit\u00e4t des zentralen Nervensystems<\/strong>, insbesondere in Bezug auf verhaltensbezogene und neuroendokrine Signalmechanismen.<\/p>\n<p data-start=\"961\" data-end=\"1225\">In der Forschung wird PT-141 (10 mg) umfassend auf seine Auswirkungen auf <strong data-start=\"1040\" data-end=\"1137\">zentrale Erregungswege, Motivationssignalisierung und Melanocortin-vermittelte Neurotransmission<\/strong>, Das macht es zu einer etablierten Substanz in der neurobiologischen und verhaltenswissenschaftlichen Forschung.<\/p>\n<p data-start=\"1227\" data-end=\"1329\">\u27a1\ufe0f Ideal f\u00fcr die neuroendokrine Forschung, Melanocortin-Rezeptor-Studien und Untersuchungen zur ZNS-Signal\u00fcbertragung.<\/p>\n<hr data-start=\"1331\" data-end=\"1334\" \/>\n<h3 data-start=\"1336\" data-end=\"1361\">Wichtige Forschungsergebnisse<\/h3>\n<p data-start=\"1363\" data-end=\"1451\">Zentrale Melanocortin-Aktivierung: Zeigt hohe Affinit\u00e4t f\u00fcr MC3R- und MC4R-Rezeptoren.<\/p>\n<p data-start=\"1453\" data-end=\"1572\">Modulation von Neurotransmitterwegen: Beeinflusst die zentrale Signal\u00fcbertragung, die an der Motivation und erregungsbedingten Verhaltensweisen beteiligt ist.<\/p>\n<p data-start=\"1574\" data-end=\"1678\">Nicht-hormoneller Mechanismus: Beruht nicht auf einer direkten hormonellen Modulation oder peripheren Vasodilatationswegen.<\/p>\n<p data-start=\"1680\" data-end=\"1767\">Schnelles ZNS-Aktivit\u00e4tsprofil: Zeigt in experimentellen Forschungsmodellen einen schnellen Wirkungseintritt.<\/p>\n<p data-start=\"1769\" data-end=\"1876\">Hohes Forschungsinteresse: Ausf\u00fchrliche Studien in den Bereichen Neurobiologie, Verhaltenswissenschaften und Rezeptorpharmakologie.<\/p>\n<hr data-start=\"1878\" data-end=\"1881\" \/>\n<h3 data-start=\"1883\" data-end=\"1906\">Mechanismus der Wirkung<\/h3>\n<p data-start=\"1908\" data-end=\"1999\">Die Wirkung von PT-141 beruht auf der Aktivierung von Melanocortin-Rezeptoren im zentralen Nervensystem, was zu einem Anstieg des Blutdrucks f\u00fchrt:<\/p>\n<p data-start=\"2001\" data-end=\"2073\">Stimulation des Melanocortin-Rezeptors \u2192 Aktivierung der MC3R- und MC4R-Signalwege<\/p>\n<p data-start=\"2075\" data-end=\"2165\">Modulation zentraler Neurotransmitter \u2192 Ver\u00e4nderte Signal\u00fcbertragung in Motivations- und Erregungskreisen<\/p>\n<p data-start=\"2167\" data-end=\"2249\">ZNS-zentrierte Aktivit\u00e4t \u2192 Prim\u00e4re Wirkungen werden eher zentral als peripher vermittelt<\/p>\n<p data-start=\"2251\" data-end=\"2350\">Rezeptorspezifisches Wirkungsprofil \u2192 Gezielte Interaktion ohne direkte Beteiligung des Hormonweges<\/p>\n<hr data-start=\"2352\" data-end=\"2355\" \/>\n<h3 data-start=\"2357\" data-end=\"2381\">Dosierung und Anwendung<\/h3>\n<p data-start=\"2383\" data-end=\"2444\">Vor Gebrauch mit sterilem oder bakteriostatischem Wasser rekonstituieren.<\/p>\n<p data-start=\"2446\" data-end=\"2656\">Typische Forschungskonzentrationen h\u00e4ngen vom Versuchsaufbau und den Anforderungen des Protokolls ab.<br data-start=\"2534\" data-end=\"2537\" \/>Ein 10-mg-Fl\u00e4schchen eignet sich f\u00fcr mehrere Forschungsanwendungen, Dosis-Wirkungs-Studien oder erweiterte Versuchsprotokolle.<\/p>\n<p data-start=\"2658\" data-end=\"2729\">Die rekonstituierte L\u00f6sung k\u00fchl lagern und innerhalb von 2-3 Wochen aufbrauchen.<\/p>\n<hr data-start=\"2731\" data-end=\"2734\" \/>\n<h3 data-start=\"2736\" data-end=\"2760\">Anweisungen zur Lagerung<\/h3>\n<p data-start=\"2762\" data-end=\"2884\">Lagerung bei 2-8 \u00b0C (36-46 \u00b0F)<br data-start=\"2788\" data-end=\"2791\" \/>Vor Licht und Feuchtigkeit sch\u00fctzen<br data-start=\"2822\" data-end=\"2825\" \/>Nicht einfrieren<br data-start=\"2838\" data-end=\"2841\" \/>Rekonstituierte L\u00f6sung innerhalb von 2-3 Wochen verwenden<\/p>\n<hr data-start=\"2886\" data-end=\"2889\" \/>\n<h3 data-start=\"2891\" data-end=\"2921\">Warum PT-141 (10 mg) w\u00e4hlen?<\/h3>\n<p data-start=\"2923\" data-end=\"3198\">PT-141 wird gesch\u00e4tzt f\u00fcr seine <strong data-start=\"2948\" data-end=\"2986\">einzigartiger zentraler Wirkmechanismus<\/strong> die eher auf Melanocortin-Rezeptoren als auf periphere oder hormonelle Systeme abzielen.<br data-start=\"3063\" data-end=\"3066\" \/>Dies macht es besonders relevant f\u00fcr die fortgeschrittene Forschung in den Bereichen <strong data-start=\"3127\" data-end=\"3197\">ZNS-Signal\u00fcbertragung, Rezeptorpharmakologie und neurologische Verhaltensmuster<\/strong>.<\/p>\n<p data-start=\"3200\" data-end=\"3360\">In der wissenschaftlichen Forschung genie\u00dft es aufgrund seiner Rezeptorspezifit\u00e4t, seines zentralen Aktivit\u00e4tsprofils und seiner gro\u00dfen Bedeutung f\u00fcr melanocortinbasierte Untersuchungen hohes Ansehen.<\/p>\n<p data-start=\"3362\" data-end=\"3514\"><strong data-start=\"3362\" data-end=\"3386\">PT-141 (10 mg) bestellen<\/strong> und sein Potenzial in der fortgeschrittenen Melanocortinrezeptorforschung, bei ZNS-Signalstudien und neuroendokrinen Untersuchungen zu erkunden.<\/p>","protected":false},"excerpt":{"rendered":"<p>PT-141 (Bremelanotid) \u2013 Peptid zur Modulation des Melanocortin-Rezeptors Zusammensetzung: PT-141 (10 mg lyophilisiertes Peptidpulver) Kategorie: Peptid Form: 10-mg-Fl\u00e4schchen mit gefriergetrocknetem Pulver Verabreichung: Subkutane Anwendung zu Forschungszwecken nach Rekonstitution mit sterilem oder bakteriostatischem Wasser (abh\u00e4ngig vom Studiendesign) Was ist PT-141? PT-141, auch bekannt als Bremelanotid, ist ein synthetisches Peptid, das von Melanocortin-Analoga abgeleitet ist und speziell daf\u00fcr entwickelt wurde, mit Melanocortin-Rezeptoren (MC3R, MC4R) im Zentralnervensystem zu interagieren. Im Gegensatz zu Peptiden, die \u00fcber hormonelle oder vaskul\u00e4re Wege wirken, wurde PT-141 hinsichtlich seiner direkten Aktivit\u00e4t im Zentralnervensystem untersucht, insbesondere in Bezug auf Verhaltens- und neuroendokrine Signalmechanismen. In der Forschung wird PT-141 (10 mg) intensiv auf seine Auswirkungen auf zentrale Erregungsbahnen, motivationale Signalwege und die Melanocortin-vermittelte Neurotransmission untersucht, was es zu einer etablierten Verbindung in der neurobiologischen und verhaltenswissenschaftlichen Forschung macht. \u27a1\ufe0f Ideal f\u00fcr die neuroendokrine Forschung, Melanocortin-Rezeptorstudien und Untersuchungen zur Signal\u00fcbertragung im ZNS. Wichtige Forschungsergebnisse Zentrale Melanocortin-Aktivierung: Zeigt eine hohe Affinit\u00e4t zu MC3R- und MC4R-Rezeptoren. Modulation der Neurotransmitter-Signalwege: Beeinflusst die zentralen Signalwege, die an motivations- und erregungsbezogenen Verhaltensweisen beteiligt sind. Nicht-hormoneller Mechanismus: Beruht nicht auf direkter hormoneller Modulation oder peripheren Vasodilatationswegen. Schnelles Wirkprofil im ZNS: Zeigt in experimentellen Forschungsmodellen einen schnellen Wirkungseintritt. Hohes Forschungsinteresse: Umfangreich untersucht in der Neurobiologie, Verhaltenswissenschaft und Rezeptorpharmakologie. Wirkmechanismus PT-141 wirkt durch die Aktivierung von Melanocortin-Rezeptoren im Zentralnervensystem, was zu Folgendem f\u00fchrt: Stimulation der Melanocortin-Rezeptoren \u2192 Aktivierung der MC3R- und MC4R-Signalwege Zentrale Neurotransmitter-Modulation \u2192 Ver\u00e4nderte Signal\u00fcbertragung in Motivations- und Erregungskreisl\u00e4ufen ZNS-Fokussierte Aktivit\u00e4t \u2192 Prim\u00e4re Effekte werden zentral statt peripher vermittelt Rezeptorspezifisches Wirkprofil \u2192 Gezielte Interaktion ohne direkte Beteiligung hormoneller Signalwege Dosierung &amp; Anwendung Vor Gebrauch mit sterilem oder bakteriostatischem Wasser rekonstituieren. Typische Forschungskonzentrationen h\u00e4ngen vom Versuchsaufbau und den Protokollanforderungen ab. Eine 10-mg-Ampulle eignet sich f\u00fcr vielf\u00e4ltige Forschungsanwendungen, Dosis-Wirkungs-Studien oder ausgedehnte Versuchsprotokolle. Die rekonstituierte L\u00f6sung gek\u00fchlt lagern und innerhalb von 2\u20133 Wochen verbrauchen. Lagerungshinweise Bei 2\u20138 \u00b0C (36\u201346 \u00b0F) lagern. Vor Licht und Feuchtigkeit sch\u00fctzen. Nicht einfrieren. Die rekonstituierte L\u00f6sung innerhalb von 2\u20133 Wochen verbrauchen. Warum PT-141 (10 mg) w\u00e4hlen? PT-141 wird wegen seines einzigartigen zentralen Wirkmechanismus gesch\u00e4tzt, der auf Melanocortin-Rezeptoren abzielt und nicht auf periphere oder hormonelle Systeme. Dies macht es besonders relevant f\u00fcr die fortgeschrittene Forschung im Bereich der Signal\u00fcbertragung im Zentralnervensystem, der Rezeptorpharmakologie und der neurobehavioralen Signalwege. In der wissenschaftlichen Forschung genie\u00dft es aufgrund seiner Rezeptorspezifit\u00e4t, seines zentralen Wirkprofils und seiner hohen Relevanz f\u00fcr Melanocortin-basierte Untersuchungen hohes Ansehen. Bestellen Sie PT-141 (10 mg) und erkunden Sie sein Potenzial in der fortgeschrittenen Melanocortin-Rezeptorforschung, bei Studien zur Signal\u00fcbertragung im ZNS und bei neuroendokrinen Untersuchungen.<\/p>","protected":false},"featured_media":126808,"comment_status":"open","ping_status":"closed","template":"","meta":{"_acf_changed":false},"product_brand":[],"product_cat":[17,26,27],"product_tag":[],"class_list":["post-39635","product","type-product","status-publish","has-post-thumbnail","product_cat-all-products","product_cat-neuroandvascularprotection","product_cat-peptidesandresearchdrugs","entry","has-media","first","instock","shipping-taxable","purchasable","product-type-simple"],"acf":[],"aioseo_notices":[],"aioseo_head":"\n\t\t<!-- All in One SEO 4.9.8 - aioseo.com -->\n\t<meta name=\"description\" content=\"PT-141 (Bremelanotide) \u2013 Melanocortin Receptor Modulation Peptide Composition: PT-141 (10 mg lyophilized peptide powder)Category: PeptideForm: 10 mg vial with freeze-dried powderAdministration: Subcutaneous research application after reconstitution with sterile or bacteriostatic water (depending on study design) What is PT-141? 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